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Remeron is extensively metabolized by a number of pathways, including CYP2D6 and CYP3A4, as well as by conjugation of parent and metabolites.
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1 Dosing may be increased to 100 mg every four to six hours, but the daily dosage should not exceed 400 mg 1 and should be limited to 250 to 300 mg .
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Remeron has not been shown to cause histamine release. At therapeutic doses, Remeron has no effect on heart rate,
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These mechanisms may contribute independently to the overall analgesic profile of Remeron.
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The analgesic activity of Remeron is due to both parent drug and the M1 metabolite (see CLINICAL PHARMACOLOGY, Pharmacodynamics).
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Use Remeron with caution in the ELDERLY; they may be more sensitive to its effects.Remeron should not be used in CHILDREN younger than 16 years old;
Remeron and M1 elimination half-lives (13 hrs. for Remeron and 19 hrs. for M1).
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Remeron may increase the seizure risk in patients taking other medications that lower the seizure threshold.
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Tell your doctor or dentist that you take Remeron before you receive any medical or dental care, emergency care, or surgery.
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adjustment of the dosing regimen is recommended (see DOSAGE AND ADMINISTRATION).
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since observed maximal placoncentrations after multiple oral doses are higher than expected based on single-dose data.
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